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Compound
PGDB_C002263
4 activity records1 related patents
2D structure
COc1ccc2nc([C@H]3CC[C@H](C(=O)Nc4cccc(CNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)c4)CC3)sc2n1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 1.51 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A028944 | PGDB_C002263 | PGDB_AS001914 | View |
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A034872 | PGDB_C002263 | PGDB_AS001555 | View |
| GI50 | - | = | 0.46 | nM | - | — | GSPT1 | - | NCI-H929 | WO2023237116A1 | PGDB_A044045 | PGDB_C002263 | PGDB_AS000710 | View |
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A061508 | PGDB_C002263 | PGDB_AS002200 | View |