Assay
PGDB_AS001914
System: cell_basedCell line: Hep3B
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 22.29 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A009004 | PGDB_C002259 | PGDB_AS001914 | View | |
| GI50 | - | = | 0.93 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A028542 | PGDB_C002217 | PGDB_AS001914 | View | |
| GI50 | - | = | 1.51 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A028944 | PGDB_C002263 | PGDB_AS001914 | View | |
| GI50 | - | = | 1.42 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A051277 | PGDB_C002262 | PGDB_AS001914 | View | |
| GI50 | - | = | 5.62 | nM | - | — | GSPT1 | - | Hep3B | WO2023237116A1 | PGDB_A062143 | PGDB_C002218 | PGDB_AS001914 | View |