Assay
PGDB_AS000219
System: cell_basedCell line: HL-60
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 9.2 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A010092 | PGDB_C002877 | PGDB_AS000219 | View | |
| IC50 | - | = | 23 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A017879 | PGDB_C002876 | PGDB_AS000219 | View | |
| IC50 | - | = | 290 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A023978 | PGDB_C002864 | PGDB_AS000219 | View | |
| IC50 | - | = | 196 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A032363 | PGDB_C002857 | PGDB_AS000219 | View | |
| IC50 | - | = | 122 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A035575 | PGDB_C002875 | PGDB_AS000219 | View | |
| IC50 | - | = | 400 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A040131 | PGDB_C002855 | PGDB_AS000219 | View | |
| IC50 | - | = | 1464 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A045325 | PGDB_C002850 | PGDB_AS000219 | View | |
| IC50 | - | = | 10 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A055804 | PGDB_C002874 | PGDB_AS000219 | View | |
| IC50 | - | = | 234 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A058400 | PGDB_C002852 | PGDB_AS000219 | View | |
| IC50 | - | > | 1000 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A066849 | PGDB_C002858 | PGDB_AS000219 | View | |
| IC50 | - | > | 1000 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A072519 | PGDB_C002872 | PGDB_AS000219 | View |