Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C003181
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(Cn4cc(Cc5ccccc5)nn4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 94 | % | - | 4 h | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A013551 | PGDB_C003181 | PGDB_AS000251 | View |
| GI50 | - | = | 23 | nM | - | — | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A019808 | PGDB_C003181 | PGDB_AS001086 | View |
| DC50 | - | = | 5.2 | nM | - | — | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A023306 | PGDB_C003181 | PGDB_AS001663 | View |
| GI50 | - | = | 36 | nM | - | — | GSPT1 | - | NCI-H1155 | WO2024222614A1 | PGDB_A048208 | PGDB_C003181 | PGDB_AS000187 | View |