Assay context summary

Assay context

23 activity records
Activity compounds and values

Activity records

23 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C003214
GI50-=22nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A007848PGDB_C003214PGDB_AS000187View
2D structure for PGDB_C003210
GI50-=39nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A009532PGDB_C003210PGDB_AS000187View
2D structure for PGDB_C003207
GI50-=10nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A017336PGDB_C003207PGDB_AS000187View
2D structure for PGDB_C003216
GI50-=19nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A023941PGDB_C003216PGDB_AS000187View
2D structure for PGDB_C003175
GI50-=50nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A027049PGDB_C003175PGDB_AS000187View
2D structure for PGDB_C003186
GI50-=14nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A036396PGDB_C003186PGDB_AS000187View
2D structure for PGDB_C003182
GI50-=42nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A036580PGDB_C003182PGDB_AS000187View
2D structure for PGDB_C003209
GI50-=78nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A042612PGDB_C003209PGDB_AS000187View
2D structure for PGDB_C003188
GI50->1000nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A042939PGDB_C003188PGDB_AS000187View
2D structure for PGDB_C003181
GI50-=36nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A048208PGDB_C003181PGDB_AS000187View
2D structure for PGDB_C003201
GI50-=18nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A048732PGDB_C003201PGDB_AS000187View
2D structure for PGDB_C003204
GI50-=11nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A050442PGDB_C003204PGDB_AS000187View
2D structure for PGDB_C003176
GI50-=7.6nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A053015PGDB_C003176PGDB_AS000187View
2D structure for PGDB_C003184
GI50-=13nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A056085PGDB_C003184PGDB_AS000187View
2D structure for PGDB_C003218
GI50-=44nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A056819PGDB_C003218PGDB_AS000187View
2D structure for PGDB_C003213
GI50-=35nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A056865PGDB_C003213PGDB_AS000187View
2D structure for PGDB_C003183
GI50-=28nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A058858PGDB_C003183PGDB_AS000187View
2D structure for PGDB_C003191
GI50-=15nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A062901PGDB_C003191PGDB_AS000187View
2D structure for PGDB_C003202
GI50-=16nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A068494PGDB_C003202PGDB_AS000187View
2D structure for PGDB_C003190
GI50-=14nM-GSPT1-NCI-H1155WO2024222614A1PGDB_A069958PGDB_C003190PGDB_AS000187View