Assay

PGDB_AS000251

System: cell_basedTarget: GSPT1Cell line: NB4
Assay context summary

Assay context

38 activity records
Assay family% Degradation
Systemcell_based
ReadoutDmax
TargetGSPT1
E3Not specified
Cell lineNB4
Technologyluminescence
Detection targetprotein_degradation
Activity compounds and values

Activity records

38 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C003217
Dmax-=125%-4 hGSPT1-NB4WO2024222614A1PGDB_A008622PGDB_C003217PGDB_AS000251View
2D structure for PGDB_C003186
Dmax-=112%-4 hGSPT1-NB4WO2024222614A1PGDB_A010052PGDB_C003186PGDB_AS000251View
2D structure for PGDB_C003181
Dmax-=94%-4 hGSPT1-NB4WO2024222614A1PGDB_A013551PGDB_C003181PGDB_AS000251View
2D structure for PGDB_C003184
Dmax-=113%-4 hGSPT1-NB4WO2024222614A1PGDB_A015376PGDB_C003184PGDB_AS000251View
2D structure for PGDB_C003196
Dmax-=16%-4 hGSPT1-NB4WO2024222614A1PGDB_A017501PGDB_C003196PGDB_AS000251View
2D structure for PGDB_C003179
Dmax-=71%-4 hGSPT1-NB4WO2024222614A1PGDB_A023945PGDB_C003179PGDB_AS000251View
2D structure for PGDB_C003201
Dmax-=96%-4 hGSPT1-NB4WO2024222614A1PGDB_A027084PGDB_C003201PGDB_AS000251View
2D structure for PGDB_C003207
Dmax-=108%-4 hGSPT1-NB4WO2024222614A1PGDB_A027329PGDB_C003207PGDB_AS000251View
2D structure for PGDB_C003185
Dmax-=28%-4 hGSPT1-NB4WO2024222614A1PGDB_A027391PGDB_C003185PGDB_AS000251View
2D structure for PGDB_C003194
Dmax-=110%-4 hGSPT1-NB4WO2024222614A1PGDB_A029828PGDB_C003194PGDB_AS000251View
2D structure for PGDB_C003188
Dmax-=31%-4 hGSPT1-NB4WO2024222614A1PGDB_A031675PGDB_C003188PGDB_AS000251View
2D structure for PGDB_C003202
Dmax-=95%-4 hGSPT1-NB4WO2024222614A1PGDB_A031707PGDB_C003202PGDB_AS000251View
2D structure for PGDB_C003208
Dmax-=46%-4 hGSPT1-NB4WO2024222614A1PGDB_A033954PGDB_C003208PGDB_AS000251View
2D structure for PGDB_C003205
Dmax-=36%-4 hGSPT1-NB4WO2024222614A1PGDB_A039519PGDB_C003205PGDB_AS000251View
2D structure for PGDB_C003197
Dmax-=49%-4 hGSPT1-NB4WO2024222614A1PGDB_A039593PGDB_C003197PGDB_AS000251View
2D structure for PGDB_C003190
Dmax-=106%-4 hGSPT1-NB4WO2024222614A1PGDB_A043069PGDB_C003190PGDB_AS000251View
2D structure for PGDB_C003182
Dmax-=93%-4 hGSPT1-NB4WO2024222614A1PGDB_A045290PGDB_C003182PGDB_AS000251View
2D structure for PGDB_C003212
Dmax-=102%-4 hGSPT1-NB4WO2024222614A1PGDB_A045567PGDB_C003212PGDB_AS000251View
2D structure for PGDB_C003191
Dmax-=107%-4 hGSPT1-NB4WO2024222614A1PGDB_A045865PGDB_C003191PGDB_AS000251View
2D structure for PGDB_C003214
Dmax-=100%-4 hGSPT1-NB4WO2024222614A1PGDB_A046316PGDB_C003214PGDB_AS000251View
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