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Compound
PGDB_C003201
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(Cn4cc(C(F)(F)c5ccc(Cl)cc5)nn4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 4.8 | nM | - | — | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A019557 | PGDB_C003201 | PGDB_AS001663 | View |
| Dmax | - | = | 96 | % | - | 4 h | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A027084 | PGDB_C003201 | PGDB_AS000251 | View |
| GI50 | - | = | 22 | nM | - | — | GSPT1 | - | NB4 | WO2024222614A1 | PGDB_A046652 | PGDB_C003201 | PGDB_AS001086 | View |
| GI50 | - | = | 18 | nM | - | — | GSPT1 | - | NCI-H1155 | WO2024222614A1 | PGDB_A048732 | PGDB_C003201 | PGDB_AS000187 | View |