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Compound
PGDB_C005766
2 activity records1 related patents
2D structure
N#Cc1c(NS(=O)(=O)C2CC2)cc(F)c(Oc2ccc3ncn(-c4cnc(N5CCN(C(=O)CN6CCC(c7ccc(N[C@H]8CCC(=O)NC8=O)cc7F)CC6)CC5)nc4)c(=O)c3c2)c1FCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | = | 9.6 | % | 10 uM | 24 h | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A027960 | PGDB_C005766 | PGDB_AS001074 | View |
| DC50 | - | = | 8.33 | nM | - | — | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A050927 | PGDB_C005766 | PGDB_AS001629 | View |