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Compound
PGDB_C005782
2 activity records1 related patents
2D structure
N#Cc1c(NS(=O)(=O)N2CCC2)ccc(F)c1Oc1ccc2ncn(-c3cnc(N4CCN(C(=O)CN5CCC(c6ccc(N[C@H]7CCC(=O)NC7=O)cc6F)CC5)CC4)nc3)c(=O)c2c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | = | 7.25 | % | 10 uM | 24 h | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A010181 | PGDB_C005782 | PGDB_AS001074 | View |
| DC50 | - | = | 16.51 | nM | - | — | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A030662 | PGDB_C005782 | PGDB_AS001629 | View |