Assay

PGDB_AS000556

System: cell_basedTarget: CDK12Cell line: MDA-MB-468
Assay context summary

Assay context

12 activity records
Assay familyviability
Systemcell_based
ReadoutIC50
TargetCDK12
E3Not specified
Cell lineMDA-MB-468
Activity compounds and values

Activity records

12 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007327
IC50->10000nM-—CDK12-MDA-MB-468CN121108130APGDB_A009020PGDB_C007327PGDB_AS000556View
2D structure for PGDB_C007164
IC50-=20.28nM-—CDK12-MDA-MB-468CN121108130APGDB_A012172PGDB_C007164PGDB_AS000556View
2D structure for PGDB_C007325
IC50-=10.11nM-—CDK12-MDA-MB-468CN121108130APGDB_A019437PGDB_C007325PGDB_AS000556View
2D structure for PGDB_C007331
IC50-=13.5nM-—CDK12-MDA-MB-468CN121108130APGDB_A020953PGDB_C007331PGDB_AS000556View
2D structure for PGDB_C007330
IC50-=36.24nM-—CDK12-MDA-MB-468CN121108130APGDB_A036721PGDB_C007330PGDB_AS000556View
2D structure for PGDB_C007335
IC50-=353.7nM-—CDK12-MDA-MB-468CN121108130APGDB_A044111PGDB_C007335PGDB_AS000556View
2D structure for PGDB_C007333
IC50->10000nM-—CDK12-MDA-MB-468CN121108130APGDB_A048055PGDB_C007333PGDB_AS000556View
2D structure for PGDB_C007332
IC50-=196.5nM-—CDK12-MDA-MB-468CN121108130APGDB_A050347PGDB_C007332PGDB_AS000556View
2D structure for PGDB_C007328
IC50-=28.26nM-—CDK12-MDA-MB-468CN121108130APGDB_A058713PGDB_C007328PGDB_AS000556View
2D structure for PGDB_C007334
IC50-=108nM-—CDK12-MDA-MB-468CN121108130APGDB_A060697PGDB_C007334PGDB_AS000556View
2D structure for PGDB_C007329
IC50-=504.2nM-—CDK12-MDA-MB-468CN121108130APGDB_A069910PGDB_C007329PGDB_AS000556View
2D structure for PGDB_C007326
IC50-=40.9nM-—CDK12-MDA-MB-468CN121108130APGDB_A070195PGDB_C007326PGDB_AS000556View
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