Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C008039
3 activity records1 related patents
2D structure
O=C1CCC(N2Cc3ccc(CNC(=O)OC4CC(c5ccccc5F)C4)cc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.025 | uM | - | — | CDK2 | - | HEK293 | WO2025043225 | PGDB_A049191 | PGDB_C008039 | PGDB_AS000366 | View |
| IC50 | - | = | 7.3 | uM | - | — | GSPT1 | - | HEK293 | WO2025043225 | PGDB_A059244 | PGDB_C008039 | PGDB_AS002508 | View |
| Dmax | - | = | 32 | % | 10 uM | 6 h | CDK2 | - | HEK293 | WO2025043225 | PGDB_A067218 | PGDB_C008039 | PGDB_AS000735 | View |