Assay

PGDB_AS000366

System: cell_basedTarget: CDK2Cell line: HEK293
Assay context summary

Assay context

26 activity records
Assay family% Degradation
Systemcell_based
ReadoutIC50
TargetCDK2
E3Not specified
Cell lineHEK293
Technologyluminescence
Detection targetprotein_degradation
Activity compounds and values

Activity records

26 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008029
IC50-=0.025uM-—CDK2-HEK293WO2025043225PGDB_A009839PGDB_C008029PGDB_AS000366View
2D structure for PGDB_C008042
IC50-=0.017uM-—CDK2-HEK293WO2025043225PGDB_A010293PGDB_C008042PGDB_AS000366View
2D structure for PGDB_C008023
IC50-=0.028uM-—CDK2-HEK293WO2025043225PGDB_A010698PGDB_C008023PGDB_AS000366View
2D structure for PGDB_C008035
IC50-=0.023uM-—CDK2-HEK293WO2025043225PGDB_A010936PGDB_C008035PGDB_AS000366View
2D structure for PGDB_C008024
IC50-=0.25uM-—CDK2-HEK293WO2025043225PGDB_A011922PGDB_C008024PGDB_AS000366View
2D structure for PGDB_C008022
IC50-=0.043uM-—CDK2-HEK293WO2025043225PGDB_A021222PGDB_C008022PGDB_AS000366View
2D structure for PGDB_C008041
IC50-=0.076uM-—CDK2-HEK293WO2025043225PGDB_A021700PGDB_C008041PGDB_AS000366View
2D structure for PGDB_C008020
IC50-=0.15uM-—CDK2-HEK293WO2025043225PGDB_A022749PGDB_C008020PGDB_AS000366View
2D structure for PGDB_C008044
IC50-=0.029uM-—CDK2-HEK293WO2025043225PGDB_A026233PGDB_C008044PGDB_AS000366View
2D structure for PGDB_C008034
IC50-=0.12uM-—CDK2-HEK293WO2025043225PGDB_A027147PGDB_C008034PGDB_AS000366View
2D structure for PGDB_C008043
IC50-=0.31uM-—CDK2-HEK293WO2025043225PGDB_A027569PGDB_C008043PGDB_AS000366View
2D structure for PGDB_C008037
IC50-=0.32uM-—CDK2-HEK293WO2025043225PGDB_A033318PGDB_C008037PGDB_AS000366View
2D structure for PGDB_C008040
IC50-=0.11uM-—CDK2-HEK293WO2025043225PGDB_A034823PGDB_C008040PGDB_AS000366View
2D structure for PGDB_C008026
IC50-=0.23uM-—CDK2-HEK293WO2025043225PGDB_A036658PGDB_C008026PGDB_AS000366View
2D structure for PGDB_C008045
IC50-=0.17uM-—CDK2-HEK293WO2025043225PGDB_A043280PGDB_C008045PGDB_AS000366View
2D structure for PGDB_C008036
IC50-=0.055uM-—CDK2-HEK293WO2025043225PGDB_A044132PGDB_C008036PGDB_AS000366View
2D structure for PGDB_C008032
IC50-=0.5uM-—CDK2-HEK293WO2025043225PGDB_A044919PGDB_C008032PGDB_AS000366View
2D structure for PGDB_C008021
IC50-=0.037uM-—CDK2-HEK293WO2025043225PGDB_A045848PGDB_C008021PGDB_AS000366View
2D structure for PGDB_C008027
IC50-=0.21uM-—CDK2-HEK293WO2025043225PGDB_A048066PGDB_C008027PGDB_AS000366View
2D structure for PGDB_C008039
IC50-=0.025uM-—CDK2-HEK293WO2025043225PGDB_A049191PGDB_C008039PGDB_AS000366View
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