Assay

PGDB_AS000735

System: cell_basedTarget: CDK2Cell line: HEK293
Assay context summary

Assay context

26 activity records
Assay family% Degradation
Systemcell_based
ReadoutDmax
TargetCDK2
E3Not specified
Cell lineHEK293
Technologyluminescence
Activity compounds and values

Activity records

26 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008029
Dmax-=40%10 uM6 hCDK2-HEK293WO2025043225PGDB_A007954PGDB_C008029PGDB_AS000735View
2D structure for PGDB_C008028
Dmax-=39%10 uM6 hCDK2-HEK293WO2025043225PGDB_A008964PGDB_C008028PGDB_AS000735View
2D structure for PGDB_C008021
Dmax-=37%10 uM6 hCDK2-HEK293WO2025043225PGDB_A010115PGDB_C008021PGDB_AS000735View
2D structure for PGDB_C008032
Dmax-=37%10 uM6 hCDK2-HEK293WO2025043225PGDB_A018884PGDB_C008032PGDB_AS000735View
2D structure for PGDB_C008044
Dmax-=43%10 uM6 hCDK2-HEK293WO2025043225PGDB_A020358PGDB_C008044PGDB_AS000735View
2D structure for PGDB_C008037
Dmax-=23%10 uM6 hCDK2-HEK293WO2025043225PGDB_A020839PGDB_C008037PGDB_AS000735View
2D structure for PGDB_C008043
Dmax-=20%10 uM6 hCDK2-HEK293WO2025043225PGDB_A021601PGDB_C008043PGDB_AS000735View
2D structure for PGDB_C008041
Dmax-=46%10 uM6 hCDK2-HEK293WO2025043225PGDB_A022178PGDB_C008041PGDB_AS000735View
2D structure for PGDB_C008031
Dmax-=25%10 uM6 hCDK2-HEK293WO2025043225PGDB_A022359PGDB_C008031PGDB_AS000735View
2D structure for PGDB_C008025
Dmax-=45%10 uM6 hCDK2-HEK293WO2025043225PGDB_A026068PGDB_C008025PGDB_AS000735View
2D structure for PGDB_C008024
Dmax-=31%10 uM6 hCDK2-HEK293WO2025043225PGDB_A037960PGDB_C008024PGDB_AS000735View
2D structure for PGDB_C008038
Dmax-=47%10 uM6 hCDK2-HEK293WO2025043225PGDB_A039807PGDB_C008038PGDB_AS000735View
2D structure for PGDB_C008034
Dmax-=29%10 uM6 hCDK2-HEK293WO2025043225PGDB_A040700PGDB_C008034PGDB_AS000735View
2D structure for PGDB_C008026
Dmax-=40%10 uM6 hCDK2-HEK293WO2025043225PGDB_A042125PGDB_C008026PGDB_AS000735View
2D structure for PGDB_C008027
Dmax-=32%10 uM6 hCDK2-HEK293WO2025043225PGDB_A043655PGDB_C008027PGDB_AS000735View
2D structure for PGDB_C008023
Dmax-=48%10 uM6 hCDK2-HEK293WO2025043225PGDB_A045637PGDB_C008023PGDB_AS000735View
2D structure for PGDB_C008022
Dmax-=36%10 uM6 hCDK2-HEK293WO2025043225PGDB_A048277PGDB_C008022PGDB_AS000735View
2D structure for PGDB_C008033
Dmax-=42%10 uM6 hCDK2-HEK293WO2025043225PGDB_A051155PGDB_C008033PGDB_AS000735View
2D structure for PGDB_C008040
Dmax-=38%10 uM6 hCDK2-HEK293WO2025043225PGDB_A052525PGDB_C008040PGDB_AS000735View
2D structure for PGDB_C008045
Dmax-=20%10 uM6 hCDK2-HEK293WO2025043225PGDB_A054596PGDB_C008045PGDB_AS000735View
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