PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Assay
PGDB_AS002508
System: cell_based
Cell line: HEK293
Assay context summary
Assay context
16 activity records
Assay family
% Degradation
System
cell_based
Readout
IC50
E3
Not specified
Cell line
HEK293
Technology
luminescence
Activity compounds and values
Activity records
16 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
9
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A012827
PGDB_C008042
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A013556
PGDB_C008036
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A015658
PGDB_C008044
PGDB_AS002508
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A015741
PGDB_C008031
PGDB_AS002508
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A021709
PGDB_C008020
PGDB_AS002508
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A030689
PGDB_C008030
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A033125
PGDB_C008043
PGDB_AS002508
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A041920
PGDB_C008034
PGDB_AS002508
View
IC50
-
=
31
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A042896
PGDB_C008023
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A051574
PGDB_C008045
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A052408
PGDB_C008038
PGDB_AS002508
View
IC50
-
=
7.3
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A059244
PGDB_C008039
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A063723
PGDB_C008040
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A068745
PGDB_C008037
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A069550
PGDB_C008041
PGDB_AS002508
View
IC50
-
=
10
uM
-
—
GSPT1
-
HEK293
WO2025043225
PGDB_A076501
PGDB_C008035
PGDB_AS002508
View