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Compound
PGDB_C009988
4 activity records1 related patents
2D structure
O=C1CC[C@H](N2Cc3c(OCc4ccc(CN5CCN6c7ccc(F)cc7OCCC6C5)cc4)cccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 65.7 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A015748 | PGDB_C009988 | PGDB_AS001792 | View |
| DC50 | - | = | 0.025 | uM | - | — | SALL4 | - | HT-1080 | WO2023025136A1 | PGDB_A024586 | PGDB_C009988 | PGDB_AS001426 | View |
| DC50 | - | = | 0.71 | nM | - | — | IKZF1 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A048017 | PGDB_C009988 | PGDB_AS001276 | View |
| Dmax | - | = | 92.9 | % | Concentration series: 0.316 nM, 10 uM | 20 h | IKZF1 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A075032 | PGDB_C009988 | PGDB_AS000619 | View |