Assay
PGDB_AS001792
System: cell_basedTarget: SALL4Cell line: HT-1080
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 63.1 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A008114 | PGDB_C009992 | PGDB_AS001792 | View | |
| Dmax | - | = | 69.7 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A011674 | PGDB_C009601 | PGDB_AS001792 | View | |
| Dmax | - | = | 46.8 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A014325 | PGDB_C009996 | PGDB_AS001792 | View | |
| Dmax | - | = | 65.7 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A015748 | PGDB_C009988 | PGDB_AS001792 | View | |
| Dmax | - | = | 49.2 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A018285 | PGDB_C010001 | PGDB_AS001792 | View | |
| Dmax | - | = | 40.9 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A020049 | PGDB_C009998 | PGDB_AS001792 | View | |
| Dmax | - | = | 46.7 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A025271 | PGDB_C010000 | PGDB_AS001792 | View | |
| Dmax | - | = | 63 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A026260 | PGDB_C009991 | PGDB_AS001792 | View | |
| Dmax | - | = | 27.8 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A032912 | PGDB_C010002 | PGDB_AS001792 | View | |
| Dmax | - | = | 72 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A048625 | PGDB_C009985 | PGDB_AS001792 | View | |
| Dmax | - | = | 44.1 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A050109 | PGDB_C009993 | PGDB_AS001792 | View | |
| Dmax | - | = | 53.1 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A057914 | PGDB_C009989 | PGDB_AS001792 | View | |
| Dmax | - | = | 75.8 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A058938 | PGDB_C009997 | PGDB_AS001792 | View | |
| Dmax | - | = | 66.6 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A060077 | PGDB_C009995 | PGDB_AS001792 | View | |
| Dmax | - | = | 69.9 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A064905 | PGDB_C009987 | PGDB_AS001792 | View | |
| Dmax | - | = | 64.2 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A071859 | PGDB_C009990 | PGDB_AS001792 | View | |
| Dmax | - | = | 45.5 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A074897 | PGDB_C009999 | PGDB_AS001792 | View | |
| Dmax | - | = | 70.4 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A075604 | PGDB_C009986 | PGDB_AS001792 | View | |
| Dmax | - | = | 68.3 | % | Concentration series: 0.316 nM, 10 uM | 20 h | SALL4 | CRBN | HT-1080 | WO2023025136A1 | PGDB_A076075 | PGDB_C009994 | PGDB_AS001792 | View |