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Compound
PGDB_C010927
4 activity records1 related patents
2D structure
CC#Cc1cnc2c(NCc3nc4ccc(F)c(F)c4[nH]3)cc(N3CCOCC3)nn12Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | > | 0.5 | uM | - | — | - | - | MDA-MB-231 | WO2025110815A1 | PGDB_A007382 | PGDB_C010927 | PGDB_AS000344 | View |
| IC50 | - | > | 0.5 | uM | - | — | CDK12 | - | - | WO2025110815A1 | PGDB_A010380 | PGDB_C010927 | PGDB_AS002095 | View |
| IC50 | - | > | 3 | uM | - | — | POLR2A | - | - | WO2025110815A1 | PGDB_A031544 | PGDB_C010927 | PGDB_AS000589 | View |
| IC50 | - | = | 0.1-0.5 | uM | - | — | CDK13 | - | - | WO2025110815A1 | PGDB_A035637 | PGDB_C010927 | PGDB_AS001146 | View |