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Compound
PGDB_C011695
3 activity records1 related patents
2D structure
COc1nc(C)ccc1-c1nnc(N[C@H]2CN(c3ccc(C4CCC(=O)NC4=O)cc3Cl)[C@@H]2C)o1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 69.5 | nM | - | — | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A019590 | PGDB_C011695 | PGDB_AS000391 | View |
| Dmax | - | = | 3.2 | % | - | 24 h | GSPT1 | - | HEK293 | WO2025224249A1 | PGDB_A026549 | PGDB_C011695 | PGDB_AS001257 | View |
| Dmax | - | = | 60.1 | % | - | 24 h | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A058070 | PGDB_C011695 | PGDB_AS002358 | View |