Assay

PGDB_AS000391

System: cell_basedTarget: CDK2Cell line: HEK293
Assay context summary

Assay context

82 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetCDK2
E3Not specified
Cell lineHEK293
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

82 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C011710
DC50-=219.2nM-—CDK2-HEK293WO2025224249A1PGDB_A008386PGDB_C011710PGDB_AS000391View
2D structure for PGDB_C011749
DC50-=24.6nM-—CDK2-HEK293WO2025224249A1PGDB_A011084PGDB_C011749PGDB_AS000391View
2D structure for PGDB_C011743
DC50-=958.9nM-—CDK2-HEK293WO2025224249A1PGDB_A013758PGDB_C011743PGDB_AS000391View
2D structure for PGDB_C011705
DC50-=154.6nM-—CDK2-HEK293WO2025224249A1PGDB_A014581PGDB_C011705PGDB_AS000391View
2D structure for PGDB_C011715
DC50-=277.2nM-—CDK2-HEK293WO2025224249A1PGDB_A014612PGDB_C011715PGDB_AS000391View
2D structure for PGDB_C011714
DC50-=273.9nM-—CDK2-HEK293WO2025224249A1PGDB_A015469PGDB_C011714PGDB_AS000391View
2D structure for PGDB_C011734
DC50-=602.3nM-—CDK2-HEK293WO2025224249A1PGDB_A015657PGDB_C011734PGDB_AS000391View
2D structure for PGDB_C011733
DC50-=577.6nM-—CDK2-HEK293WO2025224249A1PGDB_A015692PGDB_C011733PGDB_AS000391View
2D structure for PGDB_C011727
DC50-=458.5nM-—CDK2-HEK293WO2025224249A1PGDB_A017036PGDB_C011727PGDB_AS000391View
2D structure for PGDB_C011750
DC50-=26.6nM-—CDK2-HEK293WO2025224249A1PGDB_A017856PGDB_C011750PGDB_AS000391View
2D structure for PGDB_C011697
DC50-=77.9nM-—CDK2-HEK293WO2025224249A1PGDB_A018608PGDB_C011697PGDB_AS000391View
2D structure for PGDB_C011695
DC50-=69.5nM-—CDK2-HEK293WO2025224249A1PGDB_A019590PGDB_C011695PGDB_AS000391View
2D structure for PGDB_C011709
DC50-=191.2nM-—CDK2-HEK293WO2025224249A1PGDB_A020549PGDB_C011709PGDB_AS000391View
2D structure for PGDB_C011771
DC50-=55.8nM-—CDK2-HEK293WO2025224249A1PGDB_A020866PGDB_C011771PGDB_AS000391View
2D structure for PGDB_C011693
DC50-=48.4nM-—CDK2-HEK293WO2025224249A1PGDB_A022166PGDB_C011693PGDB_AS000391View
2D structure for PGDB_C011729
DC50-=523.5nM-—CDK2-HEK293WO2025224249A1PGDB_A022919PGDB_C011729PGDB_AS000391View
2D structure for PGDB_C011704
DC50-=133.2nM-—CDK2-HEK293WO2025224249A1PGDB_A024107PGDB_C011704PGDB_AS000391View
2D structure for PGDB_C011700
DC50-=106.7nM-—CDK2-HEK293WO2025224249A1PGDB_A025201PGDB_C011700PGDB_AS000391View
2D structure for PGDB_C011759
DC50-=283nM-—CDK2-HEK293WO2025224249A1PGDB_A025458PGDB_C011759PGDB_AS000391View
2D structure for PGDB_C011766
DC50-=744.5nM-—CDK2-HEK293WO2025224249A1PGDB_A026322PGDB_C011766PGDB_AS000391View
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