Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C011743
3 activity records1 related patents
2D structure
Cc1cc(C2CCC(=O)NC2=O)ccc1N1C[C@H](Nc2nnc(-c3ccc(OC(F)(F)F)cc3)o2)[C@H]1CCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 958.9 | nM | - | — | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A013758 | PGDB_C011743 | PGDB_AS000391 | View |
| Dmax | - | = | 59.3 | % | - | 24 h | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A051764 | PGDB_C011743 | PGDB_AS002358 | View |
| Dmax | - | = | 14.1 | % | - | 24 h | GSPT1 | - | HEK293 | WO2025224249A1 | PGDB_A063743 | PGDB_C011743 | PGDB_AS001257 | View |