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COc1cc(N2CCC(N(C)Cc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | HCC827 | CN116239566A | PGDB_A009843 | PGDB_C016074 | PGDB_AS000527 | View | |
| IC50 | - | < | 50 | nM | - | — | ALK | - | SR | CN116239566A | PGDB_A016674 | PGDB_C016074 | PGDB_AS001815 | View | |
| IC50 | - | < | 50 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A022029 | PGDB_C016074 | PGDB_AS002181 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A031477 | PGDB_C016074 | PGDB_AS002251 | View | |
| IC50 | - | <= | 50 | nM | - | — | - | - | CAL-62 | CN116239566A | PGDB_A034282 | PGDB_C016074 | PGDB_AS001502 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | MDA-MB-231 | CN116239566A | PGDB_A047748 | PGDB_C016074 | PGDB_AS000594 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | PC-9 | CN116239566A | PGDB_A054839 | PGDB_C016074 | PGDB_AS000139 | View | |
| IC50 | - | = | 100-500 | nM | - | — | - | - | MM.1R | CN116239566A | PGDB_A055959 | PGDB_C016074 | PGDB_AS002529 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A055974 | PGDB_C016074 | PGDB_AS002386 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | - | - | Jurkat | CN116239566A | PGDB_A077682 | PGDB_C016074 | PGDB_AS000615 | View |