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CCc1cc2c(cc1N1CCC(N3CCN(Cc4cc(F)c5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(C)(C)c1[nH]c3cc(C#N)ccc3c1C2=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A027277 | PGDB_C019613 | PGDB_AS002386 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A036389 | PGDB_C019613 | PGDB_AS002251 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | MV-4-11 | CN116239566A | PGDB_A045850 | PGDB_C019613 | PGDB_AS000843 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A073514 | PGDB_C019613 | PGDB_AS002181 | View | |
| IC50 | - | < | 50 | nM | - | — | ALK | - | SR | CN116239566A | PGDB_A076858 | PGDB_C019613 | PGDB_AS001815 | View |