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Compound
PGDB_C024202
6 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(NN4CCN(C(c5ccc(Cl)cc5)c5ccc(Cl)cc5)CC4)c(F)cc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 20-30 | % | 10 nM | 96 h | IKZF3 | - | CFPAC-1 | WO2025162225A1 | PGDB_A013378 | PGDB_C024202 | PGDB_AS000245 | View |
| % Inhibition | - | = | 10-20 | % | 10 nM | 96 h | IKZF3 | - | A375 | WO2025162225A1 | PGDB_A025083 | PGDB_C024202 | PGDB_AS001349 | View |
| % Inhibition | - | = | 30-40 | % | 10 nM | 96 h | IKZF3 | - | MV-4-11 | WO2025162225A1 | PGDB_A050032 | PGDB_C024202 | PGDB_AS001155 | View |
| % Inhibition | - | = | 50-60 | % | 500 nM | 96 h | IKZF3 | - | CFPAC-1 | WO2025162225A1 | PGDB_A053224 | PGDB_C024202 | PGDB_AS000857 | View |
| % Inhibition | - | = | 50-60 | % | 500 nM | 96 h | IKZF3 | - | A375 | WO2025162225A1 | PGDB_A055831 | PGDB_C024202 | PGDB_AS000568 | View |
| % Inhibition | - | = | 50-60 | % | 500 nM | 96 h | IKZF3 | - | MV-4-11 | WO2025162225A1 | PGDB_A071606 | PGDB_C024202 | PGDB_AS001561 | View |