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Compound
PGDB_C024474
5 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(NN4CCC5(CC4)CN(Cc4ccc(-c6ccc(Cl)cc6)cc4)C5)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 30-40 | % | 0.5 uM | - | CRBN | CRBN | - | WO2025162225A1 | PGDB_A029670 | PGDB_C024474 | PGDB_AS002133 | View |
| % Inhibition | - | = | 70-80 | % | 2 uM | - | CRBN | CRBN | - | WO2025162225A1 | PGDB_A030815 | PGDB_C024474 | PGDB_AS002540 | View |
| % Inhibition | - | = | 40-50 | % | 10 nM | 96 h | IKZF3 | - | H196 | WO2025162225A1 | PGDB_A032238 | PGDB_C024474 | PGDB_AS001140 | View |
| % Inhibition | - | = | 20-30 | % | 500 nM | 96 h | IKZF3 | - | H196 | WO2025162225A1 | PGDB_A043939 | PGDB_C024474 | PGDB_AS000866 | View |
| % Inhibition | - | > | 30 | % | 0.1 uM | - | IKZF3 | - | - | WO2025162225A1 | PGDB_A072864 | PGDB_C024474 | PGDB_AS000472 | View |