Assay context summary

Assay context

95 activity records
Activity compounds and values

Activity records

95 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C024411
% Inhibition-=60-70%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A008420PGDB_C024411PGDB_AS000866View
2D structure for PGDB_C024229
% Inhibition-=20-30%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A008534PGDB_C024229PGDB_AS000866View
2D structure for PGDB_C024221
% Inhibition-=60-70%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A009738PGDB_C024221PGDB_AS000866View
2D structure for PGDB_C024195
% Inhibition-=80-100%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A010537PGDB_C024195PGDB_AS000866View
2D structure for PGDB_C024483
% Inhibition-=50-60%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A011194PGDB_C024483PGDB_AS000866View
2D structure for PGDB_C024475
% Inhibition-=50-60%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A013134PGDB_C024475PGDB_AS000866View
2D structure for PGDB_C024579
% Inhibition-=40-50%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A013291PGDB_C024579PGDB_AS000866View
2D structure for PGDB_C024249
% Inhibition-=50-60%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A014024PGDB_C024249PGDB_AS000866View
2D structure for PGDB_C024344
% Inhibition-=50-60%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A014296PGDB_C024344PGDB_AS000866View
2D structure for PGDB_C024385
% Inhibition-=60-70%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A014313PGDB_C024385PGDB_AS000866View
2D structure for PGDB_C024194
% Inhibition-=80-100%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A015339PGDB_C024194PGDB_AS000866View
2D structure for PGDB_C024231
% Inhibition-=40-50%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A015792PGDB_C024231PGDB_AS000866View
2D structure for PGDB_C024218
% Inhibition-=60-70%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A017298PGDB_C024218PGDB_AS000866View
2D structure for PGDB_C024504
% Inhibition-=50-60%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A017355PGDB_C024504PGDB_AS000866View
2D structure for PGDB_C024574
% Inhibition-=50-60%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A017801PGDB_C024574PGDB_AS000866View
2D structure for PGDB_C024403
% Inhibition-=60-70%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A019055PGDB_C024403PGDB_AS000866View
2D structure for PGDB_C024381
% Inhibition-=40-50%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A019881PGDB_C024381PGDB_AS000866View
2D structure for PGDB_C024409
% Inhibition-=50-60%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A021289PGDB_C024409PGDB_AS000866View
2D structure for PGDB_C024208
% Inhibition-=40-50%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A021437PGDB_C024208PGDB_AS000866View
2D structure for PGDB_C024242
% Inhibition-=50-60%500 nM96 hIKZF3-H196WO2025162225A1PGDB_A021996PGDB_C024242PGDB_AS000866View