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Compound
PGDB_C024475
6 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(NN4CC5CN(Cc6ccc(-c7ccco7)s6)CC5C4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 30-40 | % | 10 nM | 96 h | IKZF3 | - | H196 | WO2025162225A1 | PGDB_A007681 | PGDB_C024475 | PGDB_AS001140 | View |
| % Inhibition | - | = | 50-60 | % | 500 nM | 96 h | IKZF3 | - | H196 | WO2025162225A1 | PGDB_A013134 | PGDB_C024475 | PGDB_AS000866 | View |
| % Inhibition | - | = | 80-100 | % | 2 uM | - | CRBN | CRBN | - | WO2025162225A1 | PGDB_A018487 | PGDB_C024475 | PGDB_AS002540 | View |
| % Inhibition | - | = | 20-30 | % | 10 nM | 96 h | IKZF3 | - | CFPAC-1 | WO2025162225A1 | PGDB_A050786 | PGDB_C024475 | PGDB_AS000245 | View |
| % Inhibition | - | = | 40-50 | % | 500 nM | 96 h | IKZF3 | - | CFPAC-1 | WO2025162225A1 | PGDB_A055807 | PGDB_C024475 | PGDB_AS000857 | View |
| % Inhibition | - | = | 70-80 | % | 0.5 uM | - | CRBN | CRBN | - | WO2025162225A1 | PGDB_A076566 | PGDB_C024475 | PGDB_AS002133 | View |