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CCc1cc2c(cc1N1CCC(N3CCN(Cc4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(C)(C)c1[nH]c3cc(C#N)ccc3c1C2=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | PC-9 | CN116239566A | PGDB_A011048 | PGDB_C025912 | PGDB_AS000139 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | HCC827 | CN116239566A | PGDB_A014523 | PGDB_C025912 | PGDB_AS000527 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | MDA-MB-231 | CN116239566A | PGDB_A032926 | PGDB_C025912 | PGDB_AS000594 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A039121 | PGDB_C025912 | PGDB_AS002181 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A045574 | PGDB_C025912 | PGDB_AS002386 | View | |
| IC50 | - | < | 50 | nM | - | — | ALK | - | SR | CN116239566A | PGDB_A063281 | PGDB_C025912 | PGDB_AS001815 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A067046 | PGDB_C025912 | PGDB_AS002251 | View |