Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C030276
9 activity records1 related patents
2D structure
Nc1nnc(-c2ccccc2O)cc1N1CC2CCC(C1)N2c1ccnc(C2CCN(Cc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)n1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-200 | nM | - | — | - | - | BT549 | WO2026061475A1 | PGDB_A000676 | PGDB_C030276 | PGDB_AS002259 | View |
| % Inhibition | - | = | 80-90 | % | 0.5 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A001177 | PGDB_C030276 | PGDB_AS000662 | View |
| IC50 | - | = | 1-5 | nM | - | — | - | - | A375 | WO2026061475A1 | PGDB_A001595 | PGDB_C030276 | PGDB_AS002441 | View |
| IC50 | - | = | 10-20 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A002620 | PGDB_C030276 | PGDB_AS000282 | View |
| % Inhibition | - | = | 90-100 | % | 2 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A005313 | PGDB_C030276 | PGDB_AS001031 | View |
| IC50 | - | = | 10-20 | nM | - | — | - | - | CFPAC-1 | WO2026061475A1 | PGDB_A079155 | PGDB_C030276 | PGDB_AS000179 | View |
| IC50 | - | = | 200-500 | nM | - | — | - | - | A549 | WO2026061475A1 | PGDB_A081699 | PGDB_C030276 | PGDB_AS000757 | View |