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CN(Cc1ccc(N2CCC(=O)NC2=O)cc1)C1CCN(c2ccc3cc(-c4ccccc4O)nnc3c2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 200-500 | nM | - | — | - | - | BT549 | WO2026061475A1 | PGDB_A003029 | PGDB_C030442 | PGDB_AS002259 | View | |
| % Inhibition | - | = | 70-80 | % | 2 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A005331 | PGDB_C030442 | PGDB_AS001031 | View | |
| IC50 | - | = | 900-1000 | nM | - | — | - | - | CFPAC-1 | WO2026061475A1 | PGDB_A006851 | PGDB_C030442 | PGDB_AS000179 | View | |
| IC50 | - | = | 20-30 | nM | - | — | - | - | H2126 | WO2026061475A1 | PGDB_A078881 | PGDB_C030442 | PGDB_AS001417 | View | |
| % Inhibition | - | = | 40-53 | % | 0.5 uM | - | CRBN | CRBN | - | WO2026061475A1 | PGDB_A081415 | PGDB_C030442 | PGDB_AS000662 | View |