Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C030841
6 activity records1 related patents
2D structure
CO[C@H]1C[C@@H](Oc2c(C)cc(-c3ccc(-c4cn(C5CCC(=O)NC5=O)c(=O)o4)c(F)c3)nc2N)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 43 | nM | - | — | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A000386 | PGDB_C030841 | PGDB_AS001885 | View |
| DC50 | - | > | 10000 | nM | - | — | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A001574 | PGDB_C030841 | PGDB_AS000910 | View |
| DC50 | - | = | 3925 | nM | - | — | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A004556 | PGDB_C030841 | PGDB_AS000302 | View |
| Dmax | - | = | 58 | % | - | 24 h | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A004770 | PGDB_C030841 | PGDB_AS000804 | View |
| Dmax | - | = | 90 | % | - | 24 h | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A005118 | PGDB_C030841 | PGDB_AS000354 | View |
| Dmax | - | = | 42 | % | - | 24 h | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A081823 | PGDB_C030841 | PGDB_AS000982 | View |