Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C030898
6 activity records1 related patents
2D structure
CNc1nc(-c2ccc(-c3cn(C4CCC(=O)NC4=O)c(=O)o3)c(F)c2)ccc1CN1CC2(CC2)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | > | 10000 | nM | - | — | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A000403 | PGDB_C030898 | PGDB_AS000302 | View |
| DC50 | - | > | 10000 | nM | - | — | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A002341 | PGDB_C030898 | PGDB_AS000910 | View |
| DC50 | - | = | 81 | nM | - | — | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A078452 | PGDB_C030898 | PGDB_AS001885 | View |
| Dmax | - | = | 46 | % | - | 24 h | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A079623 | PGDB_C030898 | PGDB_AS000804 | View |
| Dmax | - | = | 85 | % | - | 24 h | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A081346 | PGDB_C030898 | PGDB_AS000354 | View |
| Dmax | - | = | 27 | % | - | 24 h | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A081834 | PGDB_C030898 | PGDB_AS000982 | View |