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Compound
PGDB_C030917
6 activity records1 related patents
2D structure
COC1CCC2(CC1)CN(Cc1ccc(-c3ccc(-c4cn(C5CCC(=O)NC5=O)c(=O)o4)c(F)c3)nc1N)C2Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 93 | % | - | 24 h | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A000505 | PGDB_C030917 | PGDB_AS000354 | View |
| DC50 | - | = | 2471 | nM | - | — | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A002713 | PGDB_C030917 | PGDB_AS000910 | View |
| DC50 | - | = | 38 | nM | - | — | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A003490 | PGDB_C030917 | PGDB_AS001885 | View |
| DC50 | - | = | 618 | nM | - | — | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A003763 | PGDB_C030917 | PGDB_AS000302 | View |
| Dmax | - | = | 68 | % | - | 24 h | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A003782 | PGDB_C030917 | PGDB_AS000982 | View |
| Dmax | - | = | 77 | % | - | 24 h | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A081555 | PGDB_C030917 | PGDB_AS000804 | View |