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Compound
PGDB_C030974
6 activity records1 related patents
2D structure
CC1(C)CCN(Cc2cc(N)nc(-c3ccc(-c4cn(C5CCC(=O)NC5=O)c(=O)o4)c(F)c3)c2F)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 29 | nM | - | — | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A000091 | PGDB_C030974 | PGDB_AS001885 | View |
| DC50 | - | > | 10000 | nM | - | — | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A000567 | PGDB_C030974 | PGDB_AS000910 | View |
| Dmax | - | = | 64 | % | - | 24 h | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A005247 | PGDB_C030974 | PGDB_AS000804 | View |
| Dmax | - | = | 89 | % | - | 24 h | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A077959 | PGDB_C030974 | PGDB_AS000354 | View |
| DC50 | - | = | 693 | nM | - | — | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A079463 | PGDB_C030974 | PGDB_AS000302 | View |
| Dmax | - | = | 45 | % | - | 24 h | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A081230 | PGDB_C030974 | PGDB_AS000982 | View |