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Compound
PGDB_C030981
6 activity records1 related patents
2D structure
COC1CN(Cc2cc(NC3CCC3)nc(-c3ccc(-c4cn(C5CCC(=O)NC5=O)c(=O)o4)c(F)c3)c2)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 6 | nM | - | — | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A000112 | PGDB_C030981 | PGDB_AS001885 | View |
| DC50 | - | > | 10000 | nM | - | — | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A005870 | PGDB_C030981 | PGDB_AS000910 | View |
| DC50 | - | = | 419 | nM | - | — | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A006430 | PGDB_C030981 | PGDB_AS000302 | View |
| Dmax | - | = | 61 | % | - | 24 h | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A078254 | PGDB_C030981 | PGDB_AS000804 | View |
| Dmax | - | = | 92 | % | - | 24 h | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A078732 | PGDB_C030981 | PGDB_AS000354 | View |
| Dmax | - | = | 47 | % | - | 24 h | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A081457 | PGDB_C030981 | PGDB_AS000982 | View |