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Compound
PGDB_C030983
6 activity records1 related patents
2D structure
N#Cc1ccc(C2CN(Cc3cc(NC4CCC4)nc(-c4ccc(-c5cn(C6CCC(=O)NC6=O)c(=O)o5)c(F)c4)c3)C2)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 59 | % | - | 24 h | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A000439 | PGDB_C030983 | PGDB_AS000804 | View |
| DC50 | - | = | 674 | nM | - | — | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A000751 | PGDB_C030983 | PGDB_AS000910 | View |
| DC50 | - | = | 5 | nM | - | — | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A001115 | PGDB_C030983 | PGDB_AS001885 | View |
| Dmax | - | = | 58 | % | - | 24 h | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A078724 | PGDB_C030983 | PGDB_AS000982 | View |
| Dmax | - | = | 93 | % | - | 24 h | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A079689 | PGDB_C030983 | PGDB_AS000354 | View |
| DC50 | - | = | 311 | nM | - | — | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A080001 | PGDB_C030983 | PGDB_AS000302 | View |