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Compound
PGDB_C031081
6 activity records1 related patents
2D structure
CCn1nc2ccc(-c3ccc(-c4cn(C5CCC(=O)NC5=O)c(=O)o4)c(F)c3)nc2c1NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 36 | % | - | 24 h | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A000237 | PGDB_C031081 | PGDB_AS000982 | View |
| Dmax | - | = | 47 | % | - | 24 h | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A001130 | PGDB_C031081 | PGDB_AS000804 | View |
| DC50 | - | = | 165 | nM | - | — | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A001856 | PGDB_C031081 | PGDB_AS001885 | View |
| DC50 | - | > | 10000 | nM | - | — | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A004947 | PGDB_C031081 | PGDB_AS000302 | View |
| Dmax | - | = | 88 | % | - | 24 h | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A006499 | PGDB_C031081 | PGDB_AS000354 | View |
| DC50 | - | > | 10000 | nM | - | — | IKZF3 | - | Jurkat | WO2026080794A1 | PGDB_A081299 | PGDB_C031081 | PGDB_AS000910 | View |