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Compound
PGDB_C031773
4 activity records1 related patents
2D structure
O=C1CCC(c2cccc(-c3ccc(N(c4ncc(Cl)cn4)C4CC4)cc3)c2Cl)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primary T cells | WO2026114367A1 | PGDB_A002896 | PGDB_C031773 | PGDB_AS000754 | View |
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primaryT | WO2026114367A1 | PGDB_A003251 | PGDB_C031773 | PGDB_AS000152 | View |
| IC50 | - | <= | 1 | nM | - | — | VAV1 | - | primaryT | WO2026114367A1 | PGDB_A005056 | PGDB_C031773 | PGDB_AS002534 | View |
| % Degradation | - | > | 50 | % | 10 nM | - | VAV1 | - | Jurkat | WO2026114367A1 | PGDB_A079001 | PGDB_C031773 | PGDB_AS001673 | View |