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Compound
PGDB_C032001
4 activity records1 related patents
2D structure
O=C1CCC(c2cccc(-c3ccc(C#CCn4ccccc4=O)cc3)c2Cl)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 74.7 | nM | - | — | VAV1 | - | Jurkat | WO2026119120A1 | PGDB_A001687 | PGDB_C032001 | PGDB_AS001141 | View |
| Dmax | - | = | 84.2 | % | 0.08 nM | - | VAV1 | - | Jurkat | WO2026119120A1 | PGDB_A002488 | PGDB_C032001 | PGDB_AS000246 | View |
| DC50 | - | = | 45.2 | nM | - | — | VAV1 | - | - | WO2026119120A1 | PGDB_A002615 | PGDB_C032001 | PGDB_AS001984 | View |
| Dmax | - | = | 90.4 | % | 0.02 nM | - | VAV1 | - | - | WO2026119120A1 | PGDB_A081667 | PGDB_C032001 | PGDB_AS000657 | View |