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| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | ||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 2 | nM | - | — | KRAS | - | - | PGDB_A000494 | PGDB_C031999 | PGDB_AS000596 | View | |
| IC50 | - | = | 16.3 | nM | - | — | KRAS | - | SW1990 | PGDB_A001800 | PGDB_C031939 | PGDB_AS002577 | View | |
| IC50 | - | = | 2 | nM | - | — | KRAS | - | - | PGDB_A002308 | PGDB_C031999 | PGDB_AS001265 | View | |
| IC50 | - | = | 4 | nM | - | — | KRAS | - | GP5d | PGDB_A003767 | PGDB_C031939 | PGDB_AS000902 | View | |
| IC50 | - | = | 373.1 | nM | - | — | KRAS | - | LS513 | PGDB_A004243 | PGDB_C031939 | PGDB_AS002012 | View | |
| IC50 | - | = | 1 | nM | - | — | KRAS | - | - | PGDB_A005124 | PGDB_C031999 | PGDB_AS000361 | View | |
| IC50 | - | = | 2 | nM | - | — | KRAS | - | - | PGDB_A006656 | PGDB_C032000 | PGDB_AS000361 | View | |
| IC50 | - | = | 67.8 | nM | - | — | KRAS | - | NCI-H727 | PGDB_A078203 | PGDB_C031939 | PGDB_AS000308 | View | |
| IC50 | - | = | 3 | nM | - | — | KRAS | - | - | PGDB_A078378 | PGDB_C032000 | PGDB_AS001265 | View | |
| IC50 | - | > | 1000 | nM | - | — | KRAS | - | NCI-H727 | PGDB_A078969 | PGDB_C031940 | PGDB_AS000308 | View | |
| IC50 | - | = | 5 | nM | - | — | KRAS | - | - | PGDB_A079642 | PGDB_C032000 | PGDB_AS000596 | View | |
| IC50 | - | > | 1000 | nM | - | — | KRAS | - | GP5d | PGDB_A080697 | PGDB_C031940 | PGDB_AS000902 | View |