Assay context summary

Assay context

222 activity records
Activity compounds and values

Activity records

222 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000747
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A007185PGDB_C000747PGDB_AS000102View
2D structure for PGDB_C000752
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A007793PGDB_C000752PGDB_AS000102View
2D structure for PGDB_C000806
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A008740PGDB_C000806PGDB_AS000102View
2D structure for PGDB_C000782
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A009596PGDB_C000782PGDB_AS000102View
2D structure for PGDB_C000908
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A009799PGDB_C000908PGDB_AS000102View
2D structure for PGDB_C000812
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A009829PGDB_C000812PGDB_AS000102View
2D structure for PGDB_C000881
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A010364PGDB_C000881PGDB_AS000102View
2D structure for PGDB_C000903
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A010525PGDB_C000903PGDB_AS000102View
2D structure for PGDB_C000883
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A010715PGDB_C000883PGDB_AS000102View
2D structure for PGDB_C000904
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A010939PGDB_C000904PGDB_AS000102View
2D structure for PGDB_C000929
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A010981PGDB_C000929PGDB_AS000102View
2D structure for PGDB_C000822
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A011490PGDB_C000822PGDB_AS000102View
2D structure for PGDB_C000856
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A013596PGDB_C000856PGDB_AS000102View
2D structure for PGDB_C000784
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A013756PGDB_C000784PGDB_AS000102View
2D structure for PGDB_C000937
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A013978PGDB_C000937PGDB_AS000102View
2D structure for PGDB_C000749
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A014312PGDB_C000749PGDB_AS000102View
2D structure for PGDB_C000927
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A014568PGDB_C000927PGDB_AS000102View
2D structure for PGDB_C000799
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A014583PGDB_C000799PGDB_AS000102View
2D structure for PGDB_C000889
% Degradation->=20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A014671PGDB_C000889PGDB_AS000102View
2D structure for PGDB_C000960
% Degradation-=0-20%Concentration series: 500 nM, 50 nM24 hIKZF3--CN120548310APGDB_A014836PGDB_C000960PGDB_AS000102View