Assay context summary

Assay context

57 activity records
Activity compounds and values

Activity records

57 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019194
IC50-=10-50nM-IKZF3-CAL-62WO2025016359A1PGDB_A008170PGDB_C019194PGDB_AS000262View
2D structure for PGDB_C019227
IC50-<1nM-IKZF3-CAL-62WO2025016359A1PGDB_A008257PGDB_C019227PGDB_AS000262View
2D structure for PGDB_C019216
IC50-=10-50nM-IKZF3-CAL-62WO2025016359A1PGDB_A010898PGDB_C019216PGDB_AS000262View
2D structure for PGDB_C019200
IC50-=1-5nM-IKZF3-CAL-62WO2025016359A1PGDB_A013489PGDB_C019200PGDB_AS000262View
2D structure for PGDB_C019237
IC50-=5-10nM-IKZF3-CAL-62WO2025016359A1PGDB_A013894PGDB_C019237PGDB_AS000262View
2D structure for PGDB_C019191
IC50-=10-50nM-IKZF3-CAL-62WO2025016359A1PGDB_A014108PGDB_C019191PGDB_AS000262View
2D structure for PGDB_C019198
IC50-=10-50nM-IKZF3-CAL-62WO2025016359A1PGDB_A015901PGDB_C019198PGDB_AS000262View
2D structure for PGDB_C019246
IC50-=100-500nM-IKZF3-CAL-62WO2025016359A1PGDB_A017800PGDB_C019246PGDB_AS000262View
2D structure for PGDB_C019238
IC50-=100-500nM-IKZF3-CAL-62WO2025016359A1PGDB_A017940PGDB_C019238PGDB_AS000262View
2D structure for PGDB_C019219
IC50-<1nM-IKZF3-CAL-62WO2025016359A1PGDB_A018325PGDB_C019219PGDB_AS000262View
2D structure for PGDB_C019190
IC50-=10-50nM-IKZF3-CAL-62WO2025016359A1PGDB_A019361PGDB_C019190PGDB_AS000262View
2D structure for PGDB_C019254
IC50-<1nM-IKZF3-CAL-62WO2025016359A1PGDB_A024941PGDB_C019254PGDB_AS000262View
2D structure for PGDB_C019179
IC50-=50-100nM-IKZF3-CAL-62WO2025016359A1PGDB_A025573PGDB_C019179PGDB_AS000262View
2D structure for PGDB_C019201
IC50-=10-50nM-IKZF3-CAL-62WO2025016359A1PGDB_A029881PGDB_C019201PGDB_AS000262View
2D structure for PGDB_C019253
IC50-=1-5nM-IKZF3-CAL-62WO2025016359A1PGDB_A031128PGDB_C019253PGDB_AS000262View
2D structure for PGDB_C019256
IC50-=1-5nM-IKZF3-CAL-62WO2025016359A1PGDB_A033730PGDB_C019256PGDB_AS000262View
2D structure for PGDB_C019241
IC50-=100-500nM-IKZF3-CAL-62WO2025016359A1PGDB_A036689PGDB_C019241PGDB_AS000262View
2D structure for PGDB_C019178
IC50-=50-100nM-IKZF3-CAL-62WO2025016359A1PGDB_A038839PGDB_C019178PGDB_AS000262View
2D structure for PGDB_C019199
IC50-=5-10nM-IKZF3-CAL-62WO2025016359A1PGDB_A039951PGDB_C019199PGDB_AS000262View
2D structure for PGDB_C019259
IC50-=1-5nM-IKZF3-CAL-62WO2025016359A1PGDB_A040404PGDB_C019259PGDB_AS000262View