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SIMM · NJU
Assay
PGDB_AS000554
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
94 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
CDK2
E3
Not specified
Cell line
HEK293
Technology
luminescence
Detection target
protein_degradation
Activity compounds and values
Activity records
94 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
74
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A007731
PGDB_C008113
PGDB_AS000554
View
Dmax
-
=
72
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A009338
PGDB_C008054
PGDB_AS000554
View
Dmax
-
=
55
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A009347
PGDB_C008082
PGDB_AS000554
View
Dmax
-
=
67
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A009354
PGDB_C008086
PGDB_AS000554
View
Dmax
-
=
61
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A010368
PGDB_C008052
PGDB_AS000554
View
Dmax
-
=
63
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A011377
PGDB_C008124
PGDB_AS000554
View
Dmax
-
=
71
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A011963
PGDB_C008056
PGDB_AS000554
View
Dmax
-
=
72
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A012398
PGDB_C008057
PGDB_AS000554
View
Dmax
-
=
77
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A012409
PGDB_C008119
PGDB_AS000554
View
Dmax
-
=
50
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A012790
PGDB_C008114
PGDB_AS000554
View
Dmax
-
=
73
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A013440
PGDB_C008050
PGDB_AS000554
View
Dmax
-
=
62
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A013512
PGDB_C008095
PGDB_AS000554
View
Dmax
-
=
58
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A013823
PGDB_C008085
PGDB_AS000554
View
Dmax
-
=
77
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A014390
PGDB_C008081
PGDB_AS000554
View
Dmax
-
=
76
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A014736
PGDB_C008097
PGDB_AS000554
View
Dmax
-
=
72
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A016415
PGDB_C008132
PGDB_AS000554
View
Dmax
-
=
75
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A017935
PGDB_C008102
PGDB_AS000554
View
Dmax
-
=
74
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A019581
PGDB_C008094
PGDB_AS000554
View
Dmax
-
=
75
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A020307
PGDB_C008058
PGDB_AS000554
View
Dmax
-
=
72
%
10 uM
6 h
CDK2
-
HEK293
WO2025043225
PGDB_A020566
PGDB_C008074
PGDB_AS000554
View