Assay context summary

Assay context

35 activity records
Activity compounds and values

Activity records

35 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019222
IC50-=100-500nM-IKZF3-VCaPWO2025016359A1PGDB_A014368PGDB_C019222PGDB_AS000687View
2D structure for PGDB_C019200
IC50-=5-10nM-IKZF3-VCaPWO2025016359A1PGDB_A015134PGDB_C019200PGDB_AS000687View
2D structure for PGDB_C019179
IC50-=100-500nM-IKZF3-VCaPWO2025016359A1PGDB_A018441PGDB_C019179PGDB_AS000687View
2D structure for PGDB_C019223
IC50-=50-100nM-IKZF3-VCaPWO2025016359A1PGDB_A019087PGDB_C019223PGDB_AS000687View
2D structure for PGDB_C019188
IC50-=10-50nM-IKZF3-VCaPWO2025016359A1PGDB_A019424PGDB_C019188PGDB_AS000687View
2D structure for PGDB_C019218
IC50-=1-5nM-IKZF3-VCaPWO2025016359A1PGDB_A022718PGDB_C019218PGDB_AS000687View
2D structure for PGDB_C019219
IC50-=1-5nM-IKZF3-VCaPWO2025016359A1PGDB_A023241PGDB_C019219PGDB_AS000687View
2D structure for PGDB_C019216
IC50-=10-50nM-IKZF3-VCaPWO2025016359A1PGDB_A023798PGDB_C019216PGDB_AS000687View
2D structure for PGDB_C019195
IC50-=10-50nM-IKZF3-VCaPWO2025016359A1PGDB_A027362PGDB_C019195PGDB_AS000687View
2D structure for PGDB_C019201
IC50-=50-100nM-IKZF3-VCaPWO2025016359A1PGDB_A029720PGDB_C019201PGDB_AS000687View
2D structure for PGDB_C019220
IC50-=10-50nM-IKZF3-VCaPWO2025016359A1PGDB_A033217PGDB_C019220PGDB_AS000687View
2D structure for PGDB_C019221
IC50-=5-10nM-IKZF3-VCaPWO2025016359A1PGDB_A033946PGDB_C019221PGDB_AS000687View
2D structure for PGDB_C019204
IC50-=10-50nM-IKZF3-VCaPWO2025016359A1PGDB_A034385PGDB_C019204PGDB_AS000687View
2D structure for PGDB_C019177
IC50-=5-10nM-IKZF3-VCaPWO2025016359A1PGDB_A036128PGDB_C019177PGDB_AS000687View
2D structure for PGDB_C019185
IC50-=50-100nM-IKZF3-VCaPWO2025016359A1PGDB_A036447PGDB_C019185PGDB_AS000687View
2D structure for PGDB_C019196
IC50-=50-100nM-IKZF3-VCaPWO2025016359A1PGDB_A041679PGDB_C019196PGDB_AS000687View
2D structure for PGDB_C019202
IC50-=50-100nM-IKZF3-VCaPWO2025016359A1PGDB_A045728PGDB_C019202PGDB_AS000687View
2D structure for PGDB_C019212
IC50-=10-50nM-IKZF3-VCaPWO2025016359A1PGDB_A050492PGDB_C019212PGDB_AS000687View
2D structure for PGDB_C019194
IC50-=10-50nM-IKZF3-VCaPWO2025016359A1PGDB_A053444PGDB_C019194PGDB_AS000687View
2D structure for PGDB_C019214
IC50-=500-1000nM-IKZF3-VCaPWO2025016359A1PGDB_A058357PGDB_C019214PGDB_AS000687View