Assay
PGDB_AS000782
System: cell_basedCell line: AGS
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1.112 | nM | - | — | KRAS | - | AGS | CN121181579A | PGDB_A013129 | PGDB_C024617 | PGDB_AS000782 | View | |
| IC50 | - | = | 0.7981 | nM | - | — | KRAS | - | AGS | CN121181579A | PGDB_A023337 | PGDB_C024605 | PGDB_AS000782 | View | |
| IC50 | - | = | 0.6642 | nM | - | — | KRAS | - | AGS | CN121181579A | PGDB_A041343 | PGDB_C024673 | PGDB_AS000782 | View | |
| IC50 | - | = | 8.793 | nM | - | — | KRAS | - | AGS | CN121181579A | PGDB_A041884 | PGDB_C011587 | PGDB_AS000782 | View | |
| IC50 | - | = | 0.6777 | nM | - | — | KRAS | - | AGS | CN121181579A | PGDB_A067652 | PGDB_C024627 | PGDB_AS000782 | View | |
| IC50 | - | = | 1.52 | nM | - | — | KRAS | - | AGS | CN121181579A | PGDB_A068641 | PGDB_C011631 | PGDB_AS000782 | View |