Assay
PGDB_AS000885
System: cell_basedCell line: MV-4-11
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 5 | nM | - | — | - | - | MV-4-11 | WO2024032689A1 | PGDB_A012508 | PGDB_C002501 | PGDB_AS000885 | View | |
| IC50 | - | = | 10-50 | nM | - | — | - | - | MV-4-11 | WO2024032689A1 | PGDB_A015577 | PGDB_C002505 | PGDB_AS000885 | View | |
| IC50 | - | = | 24 | nM | - | — | - | - | MV-4-11 | WO2024032689A1 | PGDB_A023156 | PGDB_C002487 | PGDB_AS000885 | View | |
| IC50 | - | = | 5-10 | nM | - | — | - | - | MV-4-11 | WO2024032689A1 | PGDB_A029103 | PGDB_C002506 | PGDB_AS000885 | View | |
| IC50 | - | = | 100-500 | nM | - | — | - | - | MV-4-11 | WO2024032689A1 | PGDB_A036778 | PGDB_C002500 | PGDB_AS000885 | View | |
| IC50 | - | = | 100-500 | nM | - | — | - | - | MV-4-11 | WO2024032689A1 | PGDB_A038375 | PGDB_C002507 | PGDB_AS000885 | View | |
| IC50 | - | = | 100-500 | nM | - | — | - | - | MV-4-11 | WO2024032689A1 | PGDB_A046921 | PGDB_C002508 | PGDB_AS000885 | View |