Assay

PGDB_AS000928

System: biochemicalTarget: RAF1 | SOS1
Assay context summary

Assay context

41 activity records
Assay familybiochemical
Systembiochemical
ReadoutIC50
TargetRAF1 | SOS1
E3Not specified
OrganismHomo sapiens
TechnologyHTRF
Activity compounds and values

Activity records

41 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C011598
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A007326PGDB_C011598PGDB_AS000928View
2D structure for PGDB_C011606
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A009637PGDB_C011606PGDB_AS000928View
2D structure for PGDB_C011595
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A009952PGDB_C011595PGDB_AS000928View
2D structure for PGDB_C011601
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A011173PGDB_C011601PGDB_AS000928View
2D structure for PGDB_C011624
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A011974PGDB_C011624PGDB_AS000928View
2D structure for PGDB_C011628
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A012503PGDB_C011628PGDB_AS000928View
2D structure for PGDB_C011597
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A014259PGDB_C011597PGDB_AS000928View
2D structure for PGDB_C011592
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A015084PGDB_C011592PGDB_AS000928View
2D structure for PGDB_C011593
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A015898PGDB_C011593PGDB_AS000928View
2D structure for PGDB_C011594
IC50-=100-1000nM-—KRAS--WO2025214350A1PGDB_A016952PGDB_C011594PGDB_AS000928View
2D structure for PGDB_C011599
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A017262PGDB_C011599PGDB_AS000928View
2D structure for PGDB_C011600
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A017867PGDB_C011600PGDB_AS000928View
2D structure for PGDB_C011621
IC50-=100-1000nM-—KRAS--WO2025214350A1PGDB_A018838PGDB_C011621PGDB_AS000928View
2D structure for PGDB_C011618
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A019890PGDB_C011618PGDB_AS000928View
2D structure for PGDB_C011590
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A020533PGDB_C011590PGDB_AS000928View
2D structure for PGDB_C011630
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A021553PGDB_C011630PGDB_AS000928View
2D structure for PGDB_C011602
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A021677PGDB_C011602PGDB_AS000928View
2D structure for PGDB_C011614
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A024960PGDB_C011614PGDB_AS000928View
2D structure for PGDB_C011587
IC50-=10-100nM-—KRAS--WO2025214350A1PGDB_A025280PGDB_C011587PGDB_AS000928View
2D structure for PGDB_C011596
IC50-=1-10nM-—KRAS--WO2025214350A1PGDB_A026255PGDB_C011596PGDB_AS000928View
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