Assay context summary

Assay context

26 activity records
Activity compounds and values

Activity records

26 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001454
IC50-=23.53nM-GSPT1-NCI-H1155CN118852145APGDB_A007000PGDB_C001454PGDB_AS001039View
2D structure for PGDB_C001466
IC50-=23.1nM-GSPT1-NCI-H1155CN118852145APGDB_A007688PGDB_C001466PGDB_AS001039View
2D structure for PGDB_C001469
IC50-=21.8nM-GSPT1-NCI-H1155CN118852145APGDB_A007709PGDB_C001469PGDB_AS001039View
2D structure for PGDB_C001476
IC50-=25.4nM-GSPT1-NCI-H1155CN118852145APGDB_A009346PGDB_C001476PGDB_AS001039View
2D structure for PGDB_C001467
IC50-=11.9nM-GSPT1-NCI-H1155CN118852145APGDB_A012720PGDB_C001467PGDB_AS001039View
2D structure for PGDB_C001473
IC50-=586.2nM-GSPT1-NCI-H1155CN118852145APGDB_A012936PGDB_C001473PGDB_AS001039View
2D structure for PGDB_C001465
IC50-=25.4nM-GSPT1-NCI-H1155CN118852145APGDB_A015479PGDB_C001465PGDB_AS001039View
2D structure for PGDB_C001461
IC50-=20.28nM-GSPT1-NCI-H1155CN118852145APGDB_A019181PGDB_C001461PGDB_AS001039View
2D structure for PGDB_C001468
IC50-=5.7nM-GSPT1-NCI-H1155CN118852145APGDB_A019638PGDB_C001468PGDB_AS001039View
2D structure for PGDB_C001455
IC50-=9.23nM-GSPT1-NCI-H1155CN118852145APGDB_A020741PGDB_C001455PGDB_AS001039View
2D structure for PGDB_C001459
IC50-=10.04nM-GSPT1-NCI-H1155CN118852145APGDB_A029240PGDB_C001459PGDB_AS001039View
2D structure for PGDB_C001479
IC50-=25nM-GSPT1-NCI-H1155CN118852145APGDB_A038032PGDB_C001479PGDB_AS001039View
2D structure for PGDB_C001471
IC50-=5.3nM-GSPT1-NCI-H1155CN118852145APGDB_A043770PGDB_C001471PGDB_AS001039View
2D structure for PGDB_C001462
IC50-=26.93nM-GSPT1-NCI-H1155CN118852145APGDB_A058277PGDB_C001462PGDB_AS001039View
2D structure for PGDB_C001458
IC50-=22.48nM-GSPT1-NCI-H1155CN118852145APGDB_A060680PGDB_C001458PGDB_AS001039View
2D structure for PGDB_C001463
IC50-=7.14nM-GSPT1-NCI-H1155CN118852145APGDB_A064160PGDB_C001463PGDB_AS001039View
2D structure for PGDB_C001460
IC50-=27.87nM-GSPT1-NCI-H1155CN118852145APGDB_A064788PGDB_C001460PGDB_AS001039View
2D structure for PGDB_C001464
IC50-=510.1nM-GSPT1-NCI-H1155CN118852145APGDB_A064852PGDB_C001464PGDB_AS001039View
2D structure for PGDB_C001457
IC50-=5.95nM-GSPT1-NCI-H1155CN118852145APGDB_A066498PGDB_C001457PGDB_AS001039View
2D structure for PGDB_C001472
IC50-=75.5nM-GSPT1-NCI-H1155CN118852145APGDB_A067785PGDB_C001472PGDB_AS001039View