Assay context summary

Assay context

41 activity records
Activity compounds and values

Activity records

41 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C011597
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A007085PGDB_C011597PGDB_AS001156View
2D structure for PGDB_C011612
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A009895PGDB_C011612PGDB_AS001156View
2D structure for PGDB_C011596
IC50-=1-10nM-KRAS-SW620WO2025214350A1PGDB_A010730PGDB_C011596PGDB_AS001156View
2D structure for PGDB_C011613
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A012246PGDB_C011613PGDB_AS001156View
2D structure for PGDB_C011601
IC50-=1-10nM-KRAS-SW620WO2025214350A1PGDB_A012472PGDB_C011601PGDB_AS001156View
2D structure for PGDB_C011615
IC50-=1-10nM-KRAS-SW620WO2025214350A1PGDB_A012626PGDB_C011615PGDB_AS001156View
2D structure for PGDB_C011611
IC50-=1-10nM-KRAS-SW620WO2025214350A1PGDB_A013379PGDB_C011611PGDB_AS001156View
2D structure for PGDB_C011633
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A013860PGDB_C011633PGDB_AS001156View
2D structure for PGDB_C011587
IC50-=1-10nM-KRAS-SW620WO2025214350A1PGDB_A014502PGDB_C011587PGDB_AS001156View
2D structure for PGDB_C011639
IC50-=100-1000nM-KRAS-SW620WO2025214350A1PGDB_A015217PGDB_C011639PGDB_AS001156View
2D structure for PGDB_C011604
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A016815PGDB_C011604PGDB_AS001156View
2D structure for PGDB_C011607
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A026476PGDB_C011607PGDB_AS001156View
2D structure for PGDB_C011602
IC50-=1-10nM-KRAS-SW620WO2025214350A1PGDB_A027916PGDB_C011602PGDB_AS001156View
2D structure for PGDB_C011631
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A029804PGDB_C011631PGDB_AS001156View
2D structure for PGDB_C011616
IC50-=1-10nM-KRAS-SW620WO2025214350A1PGDB_A036435PGDB_C011616PGDB_AS001156View
2D structure for PGDB_C011620
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A038199PGDB_C011620PGDB_AS001156View
2D structure for PGDB_C011603
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A038993PGDB_C011603PGDB_AS001156View
2D structure for PGDB_C011591
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A042729PGDB_C011591PGDB_AS001156View
2D structure for PGDB_C011595
IC50-=1-10nM-KRAS-SW620WO2025214350A1PGDB_A043175PGDB_C011595PGDB_AS001156View
2D structure for PGDB_C011598
IC50-<=1nM-KRAS-SW620WO2025214350A1PGDB_A043421PGDB_C011598PGDB_AS001156View