Assay

PGDB_AS001728

System: cell_basedTarget: CDK2Cell line: HEK293T
Assay context summary

Assay context

10 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetCDK2
E3Not specified
Cell lineHEK293T
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

10 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C011110
DC50-=12.02264434617413nM-—CDK2-HEK293TWO2026064643A1PGDB_A000290PGDB_C011110PGDB_AS001728View
2D structure for PGDB_C011112
DC50-=66.06934480075964nM-—CDK2-HEK293TWO2026064643A1PGDB_A000319PGDB_C011112PGDB_AS001728View
2D structure for PGDB_C030652
DC50-=3.019951720402019nM-—CDK2-HEK293TWO2026064643A1PGDB_A001507PGDB_C030652PGDB_AS001728View
2D structure for PGDB_C030651
DC50-=21.87761623949552nM-—CDK2-HEK293TWO2026064643A1PGDB_A002618PGDB_C030651PGDB_AS001728View
2D structure for PGDB_C026003
DC50-=10nM-—CDK2-HEK293TWO2026064643A1PGDB_A005853PGDB_C026003PGDB_AS001728View
2D structure for PGDB_C030654
DC50-=0.3235936569296281nM-—CDK2-HEK293TWO2026064643A1PGDB_A006684PGDB_C030654PGDB_AS001728View
2D structure for PGDB_C025999
DC50-=3.019951720402019nM-—CDK2-HEK293TWO2026064643A1PGDB_A078614PGDB_C025999PGDB_AS001728View
2D structure for PGDB_C026001
DC50-=28.18382931264455nM-—CDK2-HEK293TWO2026064643A1PGDB_A079634PGDB_C026001PGDB_AS001728View
2D structure for PGDB_C030653
DC50-=3.981071705534969nM-—CDK2-HEK293TWO2026064643A1PGDB_A080552PGDB_C030653PGDB_AS001728View
2D structure for PGDB_C030650
DC50-=32.35936569296281nM-—CDK2-HEK293TWO2026064643A1PGDB_A080789PGDB_C030650PGDB_AS001728View
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