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SIMM · NJU
Assay
PGDB_AS001818
System: biochemical
Target: RAF1
Assay context summary
Assay context
45 activity records
Assay family
biochemical
System
biochemical
Readout
IC50
Target
RAF1
E3
Not specified
Technology
HTRF
Activity compounds and values
Activity records
45 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A007110
PGDB_C011598
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A007143
PGDB_C011590
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A010747
PGDB_C011588
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A011262
PGDB_C011629
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A012338
PGDB_C011620
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A012583
PGDB_C011605
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A012700
PGDB_C011624
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A017205
PGDB_C011615
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A018044
PGDB_C011603
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A020767
PGDB_C011607
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A021438
PGDB_C011591
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A022595
PGDB_C011630
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A022697
PGDB_C011594
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A025010
PGDB_C011625
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A026001
PGDB_C011616
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A027006
PGDB_C011610
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A028821
PGDB_C011609
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A029341
PGDB_C011592
PGDB_AS001818
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A030016
PGDB_C011626
PGDB_AS001818
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A031598
PGDB_C011596
PGDB_AS001818
View